{"title":"Muscle Relaxants","description":"Muscle relaxant medications are a class of drugs that act on the central nervous system to decrease muscle tension and reduce muscle spasms. They can be used to treat acute muscle injuries, chronic pain conditions, and other conditions that cause muscle spasms, such as multiple sclerosis and cerebral palsy. These medications work by either relaxing the muscle directly or by affecting the communication between the nerves and muscles. Some commonly used muscle relaxants include cyclobenzaprine, carisoprodol, and methocarbamol. They should only be taken under the supervision of a medical professional and can cause drowsiness and other side effects.","products":[{"product_id":"baclofen-tablets-10-mg-by-lannett","title":"Baclofen Tablets 10 mg by Lannett 100 Count (Rx)","description":"\u003cp\u003eBaclofen tablets are primarily used as muscle relaxants to alleviate muscle spasms, stiffness, and pain associated with conditions like multiple sclerosis, spinal cord injuries, or diseases. By acting on the central nervous system, Baclofen helps to relax muscles and improve mobility and overall comfort in affected individuals. It functions by inhibiting nerve signals in the spinal cord, providing effective relief from involuntary muscle contractions and enhancing the quality of life for patients with chronic muscle-related conditions.\u003c\/p\u003e\n\u003cp\u003eBaclofen Tablets 10 mg by Lannett Company are expertly formulated to offer effective relief from muscle spasticity associated with multiple sclerosis and other neurological conditions. These tablets work by targeting the central nervous system to relieve stiffness, pain, and muscle spasms, thereby improving mobility and comfort in daily activities. Trusted by healthcare professionals, Baclofen ensures consistent quality and reliability for managing symptoms related to muscle spasticity.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eProduct Details and Features:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eActive Ingredient: \u003c\/strong\u003eEach tablet contains 10 mg of Baclofen, a well-established muscle relaxant that aids in managing spasticity.\u003cbr\u003e\u003cstrong\u003eQuantity:\u003c\/strong\u003e Available in a convenient 100-count bottle, offering ease of access and consistent availability for ongoing treatment.\u003cbr\u003e\u003cstrong\u003eEfficacy:\u003c\/strong\u003e Known for its ability to effectively alleviate muscle stiffness and improve range of motion, providing a better quality of life for patients.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eMechanism of Action:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003eBaclofen is a gamma-aminobutyric acid (GABA) derivative that exerts its effects as a central nervous system (CNS) depressant. It primarily acts on the spinal cord to inhibit both monosynaptic and polysynaptic reflexes at the spinal level. By binding to GABA-B receptors, Baclofen reduces the release of excitatory neurotransmitters, leading to decreased muscle tone and spasticity.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eDirections for Use:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003e1. Initial Dosage:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eStart with a low dose as prescribed by your healthcare provider, typically beginning with a single 10 mg tablet.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eDosage may be increased gradually based on the physician's assessment and patient's response.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003e2. Administration:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eTake the tablet orally with or without food to suit personal preference or avoid stomach upset.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eIt is advisable to adhere to a consistent schedule for maximum effectiveness.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003e3. Adherence to Prescription:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eFollow the exact dosage and frequency as prescribed.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003eDo not alter the dose without consulting your healthcare provider.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eWarnings:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eWithdrawal Risks:\u003c\/strong\u003e Abrupt discontinuation may lead to withdrawal symptoms including hallucinations or seizures. Gradual reduction under medical supervision is recommended.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eOperating Machinery:\u003c\/strong\u003e May cause dizziness or drowsiness; exercise caution when driving or operating heavy machinery.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAlcohol Interaction:\u003c\/strong\u003e Avoid alcohol consumption as it can exacerbate side effects like drowsiness.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cspan style=\"text-decoration: underline;\"\u003e\u003cstrong\u003eSide Effects:\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eCommon Side Effects:\u003c\/strong\u003e Drowsiness, dizziness, weakness, and fatigue. These may lessen as your body adjusts to the medication.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eSerious Side Effects: \u003c\/strong\u003eConfusion, mood changes, seizures, or difficulty breathing. Seek immediate medical attention if these occur.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAllergic Reactions: \u003c\/strong\u003eThough rare, symptoms may include rash, itching\/swelling, severe dizziness, or trouble breathing; discontinue use and consult a medical provider if these arise.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003eBaclofen Tablets 10 mg by Lannett Company provide a reliable and effective solution for muscle spasticity, helping you regain comfort and mobility. Always use under direct medical guidance to ensure safe and optimal results.\u003c\/p\u003e","brand":"Lannett Company","offers":[{"title":"Default Title","offer_id":12256129024072,"sku":"00527-1330-01","price":29.95,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Baclofen-Tablets-10-mg-by-Lannett-00527-1330-01.jpg?v=1733411944"},{"product_id":"baclofen-tablets-10-mg-by-lannett-1000-count","title":"Baclofen Tablets 10 mg by Teva 1000 Count (Rx)","description":"\u003c!-- Microdata markup added by Google Structured Data Markup Helper. --\u003e\n\u003cp\u003eBaclofen Tablets 10 mg by Teva is a muscle relaxer and an antispastic agent. Baclofen is used to treat muscle symptoms caused by multiple sclerosis, including spasm, pain, and stiffness. Baclofen may also be used for purposes not listed in this medication guide.\u003c\/p\u003e\n\u003cp\u003eEach tablet, for oral administration, contains 10 mg baclofen. In addition, each tablet contains the following inactive ingredients: microcrystalline cellulose, pregelatinized starch, colloidal silicon dioxide, and magnesium stearate.\u003c\/p\u003e\n\u003cp class=\"First\"\u003eBaclofen tablets USP are useful for the alleviation of signs and symptoms of spasticity resulting from multiple sclerosis, particularly for the relief of flexor spasms and concomitant pain, clonus, and muscular rigidity.\u003c\/p\u003e\n\u003cp\u003ePatients should have reversible spasticity so that baclofen treatment will aid in restoring residual function. Baclofen tablets USP may also be of some value in patients with spinal cord injuries and other spinal cord diseases.\u003c\/p\u003e\n\u003cp\u003eBaclofen tablets USP are not indicated in the treatment of skeletal muscle spasm resulting from rheumatic disorders.\u003c\/p\u003e\n\u003cp\u003eThe efficacy of baclofen in stroke, cerebral palsy, and Parkinson's disease has not been established and, therefore, it is not recommended for these conditions.\u003c\/p\u003e\n\u003cp\u003eBrand: Teva Pharmaceuticals\u003cbr\u003e\u003c\/p\u003e\n\u003cp\u003eSize: 1000 Tablets\u003cbr\u003eStrength: 10 mg\u003cbr\u003eNDC: \u003cspan data-mce-fragment=\"1\"\u003e00172-4096-80\u003c\/span\u003e\u003cbr\u003eUPC: \u003cspan data-mce-fragment=\"1\"\u003e301724096806\u003c\/span\u003e\u003c\/p\u003e\n\u003cp\u003eBuy Baclofen Tablets 10 mg by Teva\u003cspan\u003e \u003c\/span\u003e\u003cspan data-mce-fragment=\"1\"\u003emuscle relaxer to treat muscle symptoms caused by multiple sclerosis, including spasm, pain, and stiffness \u003c\/span\u003eat Mountainside Medical Equipment.\u003c\/p\u003e\n\u003c!-- Microdata markup added by Google Structured Data Markup Helper. --\u003e","brand":"Teva Pharmaceuticals","offers":[{"title":"Default Title","offer_id":12256150028360,"sku":"00172-4096-80","price":176.5,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/products\/BaclofenTablets00172-4096-80.jpg?v=1680871013"},{"product_id":"baclofen-tablets-20-mg-by-qualitest-100-count","title":"Baclofen Tablets 20 mg by Teva 100 Count (Rx)","description":"\u003c!-- Microdata markup added by Google Structured Data Markup Helper. --\u003e\n\u003cp\u003eBaclofen Tablets 20 mg by Teva a muscle relaxer and an antispastic agent. Baclofen is used to treat muscle symptoms caused by multiple sclerosis, including spasm, pain, and stiffness. Baclofen may also be used for purposes not listed in this medication guide.\u003c\/p\u003e\n\u003cp\u003e\u003cspan\u003eEach tablet, for oral administration, contains 20 mg baclofen, USP. In addition, each tablet contains the following inactive ingredients: anhydrous lactose, colloidal silicon dioxide, dibasic calcium phosphate dihydrate, magnesium stearate, microcrystalline cellulose and sodium starch glycolate.\u003c\/span\u003e\u003c\/p\u003e\n\u003cp class=\"First\"\u003eBaclofen tablets are useful for the alleviation of signs and symptoms of spasticity resulting from multiple sclerosis, particularly for the relief of flexor spasms and concomitant pain, clonus, and muscular rigidity.\u003c\/p\u003e\n\u003cp\u003ePatients should have reversible spasticity so that baclofen treatment will aid in restoring residual function. Baclofen tablets may also be of some value in patients with spinal cord injuries and other spinal cord diseases.\u003c\/p\u003e\n\u003cp\u003eBaclofen tablets are not indicated in the treatment of skeletal muscle spasm resulting from rheumatic disorders.\u003c\/p\u003e\n\u003cp\u003eThe efficacy of baclofen in stroke, cerebral palsy, and Parkinson’s disease has not been established and, therefore, it is not recommended for these conditions.\u003c\/p\u003e\n\u003cp\u003e \u003c\/p\u003e\n\u003cp\u003eBrand: Teva Pharmaceuticals\u003cbr\u003eSize: 100 Tablets\u003cbr\u003eStrength: 20 mg\u003cbr\u003eNDC: 00172-4097-60\u003cbr\u003eUPC: 301724097605\u003c\/p\u003e\n\u003cp\u003e\u003cbr\u003e\u003c\/p\u003e\n\u003cp\u003eBuy Baclofen Tablets 20 mg by Teva used to treat muscle symptoms caused by multiple sclerosis at Mountainside Medical Equipment.\u003c\/p\u003e\n\u003c!-- Microdata markup added by Google Structured Data Markup Helper. --\u003e","brand":"Teva Pharmaceuticals","offers":[{"title":"Default Title","offer_id":12256150290504,"sku":"00172-4097-60","price":26.3,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Baclofen-Tablets-20-mg-Teva-Pharmaceuticals--00172-4097-60.jpg?v=1764764558"},{"product_id":"quelicin-succinylcholine-chloride-injection-usp-20mg-ml-multi-dose-vial-10-ml-x-25-box","title":"Quelicin (Succinylcholine Chloride Injection USP) 20mg\/mL Multi-Dose Vial 10 mL x 25\/Box **Refrigerated Item","description":"\u003cp\u003eQuelicin (Succinylcholine Chloride Injection) is a muscle relaxant used during surgeries or mechanical ventilation to facilitate intubation and ensure optimal conditions for surgical procedures. It acts quickly by depolarizing neuromuscular blockers to induce short-term paralysis. This medication is essential for skilled healthcare professionals in emergency settings for rapid sequence induction and tracheal intubation. It is vital for critical patient management, ensuring controlled muscle relaxation during medical interventions.\u003c\/p\u003e\n\u003cp\u003eQuelicin (Succinylcholine Chloride Injection, USP) is a sterile, nonpyrogenic solution used as a short-acting neuromuscular blocker for intravenous administration. It is supplied in a concentration of 20 mg\/mL in multi-dose vials. The pack contains 25 vials, each having a 10 mL capacity.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eDetails and Features:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eConcentration:\u003c\/strong\u003e 20 mg\/mL of succinylcholine chloride.\u003cbr\u003e\u003cstrong\u003eFormulation: \u003c\/strong\u003eMulti-dose vials, ensuring versatility in dosing requirements.\u003cbr\u003e\u003cstrong\u003ePackaging: \u003c\/strong\u003e25 vials per box, suitable for bulk medical settings.\u003cbr\u003e\u003cstrong\u003eAdministration Route:\u003c\/strong\u003e Intravenous use for rapid onset action.\u003cbr\u003e\u003cstrong\u003eIndication: \u003c\/strong\u003eQuelicin is primarily used to facilitate tracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eMechanism of Action:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003eSuccinylcholine is a depolarizing neuromuscular blocker. It mimics the action of acetylcholine, binding to nicotinic receptors at the neuromuscular junction. This binding results in depolarization of the muscle endplate, leading initially to muscle fasciculations followed by paralysis. Its action is terminated by the rapid hydrolysis of succinylcholine by plasma cholinesterases, resulting in a brief duration of action.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eWarnings:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eMalignant Hyperthermia:\u003c\/strong\u003e Succinylcholine may trigger this genetic disorder, characterized by a rapid increase in body temperature and severe muscle contractions. Early recognition and treatment with dantrolene is essential.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eHyperkalemia Risk:\u003c\/strong\u003e Can cause significant potassium release, resulting in potentially life-threatening hyperkalemia, especially in patients with burns, neurological disorders, or muscle trauma.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eCardiac Arrest: \u003c\/strong\u003eRare cases have been reported in children, typically associated with undiagnosed neuromuscular disorders.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eProlonged Paralysis\u003c\/strong\u003e: May occur in individuals with atypical plasma cholinesterase or other conditions affecting metabolism or excretion.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAnaphylaxis:\u003c\/strong\u003e As with other neuromuscular blockers, potential for severe allergic reactions exists.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cspan style=\"text-decoration: underline;\"\u003e\u003cstrong\u003eSide Effects:\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eMuscle Fasciculations: \u003c\/strong\u003eVisible muscle twitches prior to paralysis.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eBradycardia or Tachycardia:\u003c\/strong\u003e Changes in heart rate can occur post-administration.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eIncreased Intraocular Pressure: \u003c\/strong\u003eMay transiently increase eye pressure.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eMyoglobinemia\/Myoglobinuria:\u003c\/strong\u003e Rhabdomyolysis can occur.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eProlonged Apnea:\u003c\/strong\u003e Particularly in cases of pseudocholinesterase deficiency.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eClinical Consideration:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eMonitoring: \u003c\/strong\u003eUse with appropriate monitoring of neuromuscular function, especially in settings lacking emergency equipment.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003ePatient History:\u003c\/strong\u003e Thorough assessment of the patient's medical history and potential risk factors for complications is necessary before administration.\u003cbr\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eResuscitation Equipment:\u003c\/strong\u003e Immediate availability of resuscitative drugs and equipment is mandatory when using this medication.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003eAlways consult the prescribing information and a healthcare professional for comprehensive details and specific clinical use cases.\u003c\/p\u003e","brand":"Pfizer Injectables","offers":[{"title":"Default Title","offer_id":39953372151880,"sku":"00409-6629-02","price":1255.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Quelicin-_Succinylcholine-Chloride-Injection-USP-20mg-mL.jpg?v=1684860935"},{"product_id":"baclofen-usp-for-compounding-api","title":"Baclofen USP For Compounding (API)  (Rx)","description":"\u003cp\u003eBaclofen USP active pharmaceutical ingredient (API) is a centrally acting muscle relaxant that is used to treat symptoms of spastic movement disorders, such as multiple sclerosis, spinal cord injury, or cerebral palsy. It is a derivative of gamma-aminobutyric acid (GABA), a neurotransmitter in the brain that plays a role in regulating muscle tone. Baclofen works by binding to specific GABA receptors, reducing the activity of neurons that cause muscle spasms and stiffness. It is considered a safe and effective treatment, with minimal side effects, for spasticity.\u003c\/p\u003e\n\u003cp\u003e\u003cspan style=\"color: rgb(255, 42, 0);\"\u003e\u003cstrong\u003eShips in 2-4 business days.\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cp\u003eBaclofen USP  is a muscle relaxant medication commonly used for the treatment of muscle spasticity due to conditions such as multiple sclerosis, cerebral palsy, or spinal cord injuries. It may also be prescribed for other conditions that cause muscle spasms such as chronic low back pain or migraines. Baclofen USP may be used for compounding, meaning it can be formulated into different dosage forms such as creams, ointments, gels, or transdermal patches, to meet specific patient needs or preferences. Compounding can also allow for customized strengths or combinations of medications, which may be beneficial for certain patients who may not respond well to commercially available products. However, it is important to note that the use of compounded medications should be discussed with a physician and only obtained from a reputable compounding pharmacy.\u003c\/p\u003e","brand":"Mountainside Medical","offers":[{"title":"25 g","offer_id":40071594213448,"sku":"3209-04","price":145.0,"currency_code":"USD","in_stock":true},{"title":"100 g","offer_id":40071594246216,"sku":"3209-05","price":490.0,"currency_code":"USD","in_stock":true},{"title":"500 g","offer_id":40071594278984,"sku":"3209-08","price":1975.0,"currency_code":"USD","in_stock":true},{"title":"1 Kg","offer_id":40071594311752,"sku":"3209-09","price":2950.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Baclofen-USP-For-Compounding-_API.jpg?v=1706707190"},{"product_id":"methocarbamol-usp-for-compounding-api","title":"Methocarbamol USP For Compounding (API)","description":"\u003cp\u003eMethocarbamol USP For Compounding (API) is a high-quality active pharmaceutical ingredient used in the formulation of medications aimed at providing muscle relaxation and pain relief. It is commonly used to treat musculoskeletal conditions such as muscle spasms, strains, and sprains. Methocarbamol works by depressing the central nervous system, leading to muscle relaxation and alleviating discomfort associated with acute musculoskeletal disorders. This API enables healthcare professionals to compound personalized therapies, optimizing treatment effectiveness and patient care. Key health-related benefits include enhanced recovery from injuries, improved mobility, and a reduction in muscle-related pain, making it integral to pain management and orthopedic care.\u003c\/p\u003e\n\u003cp\u003e\u003cspan style=\"color: rgb(255, 42, 0);\"\u003e\u003cstrong\u003eShips in 2-4 business days.\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cp\u003eMethocarbamol USP is a medication used for its muscle relaxant properties. It is often used in compounding pharmacies to create customized medication formulations for patients who may have specific needs or preferences. It is made of methocarbamol, an active ingredient, and other inactive ingredients such as binders, fillers, and preservatives. These additional ingredients may vary depending on the specific formulation and needs of the patient. Methocarbamol USP is available in a variety of dosage forms including tablets, capsules, and injectables.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eCAS Number: 532-03-06\u003cbr\u003e\u003c\/strong\u003e\u003c\/p\u003e","brand":"Mountainside Medical","offers":[{"title":"100 g","offer_id":40078634090568,"sku":"1943-05","price":62.0,"currency_code":"USD","in_stock":true},{"title":"500 g","offer_id":40078634123336,"sku":"1943-08","price":195.0,"currency_code":"USD","in_stock":true},{"title":"1 Kg","offer_id":40078634156104,"sku":"1943-09","price":329.0,"currency_code":"USD","in_stock":true},{"title":"5 Kg","offer_id":40078634188872,"sku":"1943-03","price":1295.0,"currency_code":"USD","in_stock":true},{"title":"20 Kg","offer_id":40078634221640,"sku":"1943-06","price":4400.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Methocarbamol-USP-For-Compounding-_API_-_Rx.jpg?v=1706727137"},{"product_id":"tizanidine-hydrochloride-usp-for-compounding-api","title":"Tizanidine Hydrochloride USP For Compounding (API)","description":"\u003cp\u003eTimolol Maleate USP for Compounding (API) is an active pharmaceutical ingredient used to formulate ophthalmic solutions and other medications for treating glaucoma and ocular hypertension. As a non-selective beta-blocker, it reduces intraocular pressure by decreasing the production of aqueous humor in the eye, helping prevent optic nerve damage and vision loss. Compounding pharmacists prepare customized doses tailored to specific patient needs, ensuring effective management of these conditions while minimizing side effects and maximizing therapeutic benefits.\u003c\/p\u003e\n\u003cp\u003e\u003cspan style=\"color: rgb(255, 42, 0);\"\u003e\u003cstrong\u003eShips in 2-4 business days.\u003c\/strong\u003e\u003c\/span\u003e\u003c\/p\u003e\n\u003cp\u003eTizanidine Hydrochloride USP is a medication used for compounding that is used to treat muscle spasms and muscle tightness caused by conditions such as multiple sclerosis or spinal cord injury. It is a muscle relaxant that can help reduce pain and improve mobility in affected individuals. When compounded, it can be made into different forms such as creams, gels, or ointments for topical application, or into suspensions for oral administration. Compounding allows for personalized dosing and delivery methods, making it a useful option for patients who may have difficulty swallowing pills or need a specific strength or form of the medication.\u003c\/p\u003e\n\u003cp\u003eTizanidine hydrochloride USP active pharmaceutical ingredient (API) is a prescription medication used to treat muscle spasms and increased muscle tone caused by conditions such as multiple sclerosis, spinal cord injury, or other neurological disorders. It works by acting on certain nerve cells in the spinal cord to suppress abnormal nerve impulses that cause muscle spasticity.\u003cbr\u003e\u003cbr\u003eTizanidine hydrochloride is a centrally acting muscle relaxant and belongs to the class of drugs known as alpha-2 adrenergic agonists. It is sold under the brand name Zanaflex and is available in oral tablet and capsule forms.\u003cbr\u003e\u003cbr\u003eAs an API, tizanidine hydrochloride is the active chemical component responsible for the therapeutic effects of the medication. It is used to develop various formulations and dosage forms of tizanidine for administration to patients. API is the primary ingredient that makes a medication effective in treating a specific medical condition.\u003cbr\u003e\u003cbr\u003e\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eCAS Number: 64461-82-1\u003c\/strong\u003e\u003cbr\u003e\u003c\/p\u003e","brand":"Mountainside Medical","offers":[{"title":"25 g","offer_id":40079577874504,"sku":"2351-04","price":875.0,"currency_code":"USD","in_stock":true},{"title":"100 g","offer_id":40079577907272,"sku":"2351-05","price":2750.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Tizanidine_Hydrochloride_USP_For_Compounding_API.jpg?v=1729691325"},{"product_id":"dantrium-dantrolene-sodium-capsules-25-mg-100-bottle-rx","title":"Dantrium (Dantrolene Sodium) Capsules 25 mg, 100\/Bottle (RX)","description":"\u003cp\u003eDANTRIUM (dantrolene) is a muscle relaxant that is used to treat muscle spasms and stiffness caused by conditions such as cerebral palsy, multiple sclerosis, and spinal cord injuries. It may also be used during anesthesia to prevent or reduce muscle contractions during surgery. In some cases, it may also be prescribed for the treatment of a rare genetic condition called malignant hyperthermia that causes a severe increase in body temperature and muscle rigidity.\u003c\/p\u003e\n\u003cp\u003eDantrium (dantrolene sodium) capsules 25 mg is a prescription medication used to treat muscle spasms caused by conditions such as spinal cord injury, stroke, cerebral palsy, multiple sclerosis, or other conditions affecting the muscles. It works by relaxing the muscles and preventing the release of substances that cause muscle contractions. This medication is available in capsule form and is usually taken three times a day as directed by a doctor. It is usually used in combination with physical therapy and other treatments to help improve muscle control and function. Common side effects may include drowsiness, dizziness, weakness, nausea, diarrhea, and difficulty breathing. It is important to talk to a doctor before taking this medication, as it may interact with other medications or have adverse effects in people with certain medical conditions.\u003c\/p\u003e\n\u003cp\u003eDantrium (Dantrolene Sodium) Capsules 25 mg work by suppressing the release of calcium from muscle cells, which leads to relaxation of the muscle. This mechanism of action is thought to occur by binding to specific receptors on the surface of muscle cells called ryanodine receptors.\u003c\/p\u003e\n\u003cp\u003eThese receptors are involved in regulating the levels of calcium inside muscle cells. Normally, when a signal from the nerve reaches the muscle, calcium is released inside the muscle cell, which causes it to contract.\u003c\/p\u003e\n\u003cp\u003eIn certain disorders such as spasticity or malignant hyperthermia, there is an excessive release of calcium in the muscle cells, causing prolonged or uncontrollable muscle contractions. 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This action reduces muscle contraction and spasticity.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eDirections:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eTake the medication as prescribed by your healthcare provider.\u003c\/li\u003e\n\u003cli\u003eSwallow capsules whole with a full glass of water.\u003c\/li\u003e\n\u003cli\u003eMay be taken with or without food.\u003c\/li\u003e\n\u003cli\u003eDo not alter dosage without consulting your doctor.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eWarnings:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eUse with caution in patients with liver disease due to risk of liver toxicity.\u003c\/li\u003e\n\u003cli\u003eRegular liver function tests may be required during treatment.\u003c\/li\u003e\n\u003cli\u003eInform your healthcare provider of all medications and supplements you are using to avoid interactions.\u003c\/li\u003e\n\u003cli\u003eNot recommended for situations requiring fine motor control.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cstrong\u003eSide Effects:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cp\u003eCommon side effects include:\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eDrowsiness\u003c\/li\u003e\n\u003cli\u003eWeakness\u003c\/li\u003e\n\u003cli\u003eDizziness\u003c\/li\u003e\n\u003cli\u003eDiarrhea\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003eSeek immediate medical attention if you experience:\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003eSigns of liver problems (yellowing of skin or eyes, dark urine)\u003c\/li\u003e\n\u003cli\u003eSevere fatigue\u003c\/li\u003e\n\u003cli\u003eDifficulty swallowing or breathing\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003eDantrolene Sodium Capsules by Amneal Pharmaceuticals provide a reliable solution for managing muscle spasticity, improving mobility and comfort. 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Trust the proven, doctor-recommended muscle relaxer that delivers safe and effective results so you can regain comfort and confidence in your daily life.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eOrder today and start your journey to better movement and muscle relaxation—backed by Advagen Pharma’s commitment to your health.\u003c\/strong\u003e\u003c\/p\u003e","brand":"Advagen Pharma","offers":[{"title":"Default Title","offer_id":53189656510832,"sku":"72888-0009-01","price":23.95,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Baclofen-Tablets-5-mg-by-Advagen-100-Count.jpg?v=1768831386"},{"product_id":"papaverine-hydrochloride-injection-60-mg-2ml-oryza-pharmaceutical-72516-0024-10","title":"Papaverine Hydrochloride Injection 60 mg\/2mL Single Dose Vials 2 mL x 10\/Box (RX)","description":"\u003ch1\u003eVasodilator \u0026amp; Smooth Muscle Relaxant\u003c\/h1\u003e\n\u003cp\u003ePapaverine Hydrochloride 60mg\/2mL is a \u003cstrong\u003eprescription-strength injectable medication\u003c\/strong\u003e formulated to relax smooth muscles and dilate blood vessels. Each sterile 2 mL single-dose vial contains \u003cstrong\u003e60 mg of Papaverine HCl\u003c\/strong\u003e (30 mg\/mL), providing a ready-to-use injectable solution. Administered only by healthcare professionals (intramuscularly or via slow IV infusion), Papaverine injection is used to \u003cstrong\u003eimprove circulation and relieve muscle spasms\u003c\/strong\u003e in various medical conditions. Its potent vasodilator action makes it ideal for treating \u003cstrong\u003eerectile dysfunction (ED)\u003c\/strong\u003e, \u003cstrong\u003eperipheral and cerebral vascular spasms\u003c\/strong\u003e, and \u003cstrong\u003evisceral smooth muscle cramps\u003c\/strong\u003e.\u003c\/p\u003e\n\u003ch2\u003eUses\u003c\/h2\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003ePowerful Vasodilator \u0026amp; Spasmolytic:\u003c\/strong\u003e Papaverine directly relaxes smooth muscles in blood vessels and organs, increasing circulation. It is classified as a \u003cstrong\u003edirect-acting vasodilator\u003c\/strong\u003e (benzylisoquinoline alkaloid).\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eIndicated for ED and Vascular Disorders:\u003c\/strong\u003e Clinically used to treat male ED by increasing penile blood flow, and to relieve arterial spasms in peripheral vascular disease, Raynaud’s phenomenon, and cerebral vasospasm. It can also ease \u003cstrong\u003evisceral muscle spasms\u003c\/strong\u003e in the gastrointestinal or biliary tract.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eIntracavernosal Injection Therapy:\u003c\/strong\u003e For erectile dysfunction, Papaverine is often injected directly into the penis (intracavernosal) – sometimes in combination with phentolamine or prostaglandin – to induce a firm erection. Unlike oral ED drugs, this method works locally and can be effective when other treatments fail.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eSingle-Dose Sterile Vials:\u003c\/strong\u003e Each glass ampoule contains a clear, colorless solution of Papaverine HCl. The amber-colored 2 mL vial ensures drug stability. Being single-use, it minimizes contamination – simply dispose after one injection.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAdministration:\u003c\/strong\u003e Supplied in ready-to-use injectable form. Papaverine is given via \u003cstrong\u003eintramuscular (IM) or slow intravenous (IV)\u003c\/strong\u003e injection. It \u003cstrong\u003emust be injected slowly\u003c\/strong\u003e (over 1–2 minutes) to avoid rapid drops in blood pressure or heart arrhythmias. All doses and frequency are determined by a doctor based on the patient’s condition.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003ePrescription Only:\u003c\/strong\u003e This medication requires a doctor’s prescription and oversight. It should \u003cem\u003enever\u003c\/em\u003e be self-administered without proper training. Under supervision, Papaverine can be an effective therapy for improving circulation.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch2\u003eComposition \u0026amp; Formulation\u003c\/h2\u003e\n\u003cp\u003eEach 2 mL ampoule of Papaverine Injection contains:\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eActive ingredient:\u003c\/strong\u003e 60 mg Papaverine Hydrochloride (30 mg per 1 mL). Papaverine is a vasodilating smooth-muscle relaxant derived synthetically or from opium.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eExcipients:\u003c\/strong\u003e Includes 0.45 mg disodium EDTA per ampoule as a stabilizer. The solution is sterile, pyrogen-free, and preservative-free.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eForm:\u003c\/strong\u003e A clear, colorless injectable solution in an amber glass ampoule. The 2 mL single-dose format ensures accurate dosing and sterility.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch2\u003eHow It Works (Mechanism of Action)\u003c\/h2\u003e\n\u003cp\u003ePapaverine’s primary action is \u003cstrong\u003edirect spasmolysis of smooth muscle\u003c\/strong\u003e. It works by inhibiting the contractility of vascular and visceral muscles, leading to vessel dilation and muscle relaxation. Key points of its mechanism:\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eVasodilation:\u003c\/strong\u003e Papaverine acts most strongly on arterial smooth muscle. It relaxes coronary, cerebral, pulmonary and peripheral arteries, markedly increasing blood flow to these regions. For example, dilation of penile arteries enables erection, while relaxation of cerebral vessels can improve brain perfusion.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eSmooth Muscle Relaxation:\u003c\/strong\u003e Beyond vessels, Papaverine relaxes \u003cstrong\u003ebronchial, gastrointestinal, ureteral, and biliary\u003c\/strong\u003e smooth muscle. This helps relieve spasms in the intestines or biliary tract (e.g. intestinal cramp or gallbladder colic).\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eCardiac Effects:\u003c\/strong\u003e It also mildly depresses cardiac excitability and prolongs myocardial refractory period. Although no longer first-line for heart issues, it has been used in certain arrhythmias and angina when other drugs are unsuitable.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eEnhanced Collateral Flow:\u003c\/strong\u003e In cases of arterial blockage, Papaverine may reduce reflex vasoconstriction in collateral vessels, improving blood supply to ischemic tissues.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003eThrough these actions, Papaverine injection helps \u003cstrong\u003eincrease oxygen delivery and relieve pain related to spasms\u003c\/strong\u003e. Its combined vasodilator and spasmolytic effects make it valuable in circulatory disorders and muscle cramp conditions.\u003c\/p\u003e\n\u003ch2\u003eIndications and Benefits\u003c\/h2\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eErectile Dysfunction (ED):\u003c\/strong\u003e Papaverine 60mg injection is an established therapy for ED. By relaxing penile smooth muscle, it enhances penile blood flow and induces an erection usable for sexual intercourse. It is especially helpful when oral ED medications are ineffective or contraindicated. In practice, one 2 mL dose is injected into the penis under medical supervision. Many men experience firmer erections and improved sexual performance without systemic side effects of oral drugs.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003ePeripheral Vascular Disease (PVD):\u003c\/strong\u003e In conditions like peripheral artery disease or Raynaud’s phenomenon, narrowed arteries reduce limb blood flow. Papaverine injection relaxes these peripheral arteries, improving circulation to the arms and legs. Patients often report relief from symptoms like leg cramps, numbness, or cold extremities after therapy.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eCerebral Arterial Spasm:\u003c\/strong\u003e Papaverine can be used to counteract cerebral vasospasm (e.g., after subarachnoid hemorrhage or head injury). By dilating cerebral arteries, it helps restore brain perfusion. In neurosurgery settings, Papaverine infusion has been used to prevent or treat arterial spasms, potentially reducing stroke risk.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eVisceral Spasms:\u003c\/strong\u003e Smooth muscle cramps in the gastrointestinal (GI) tract, bile ducts or ureters can cause severe pain. Papaverine’s action on GI and biliary smooth muscle means it can relieve such spasms. For instance, in biliary colic or intestinal cramping (colitis, irritable bowel), Papaverine injection or infusion provides muscular relaxation and pain relief.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eOther Uses:\u003c\/strong\u003e Historically, Papaverine was trialed in angina and hypertension, though it is now superseded by better drugs. It has utility in certain heart rhythm disorders by relaxing cardiac muscle. Its broad smooth-muscle relaxant effect also means it can be used off-label for conditions involving involuntary muscle contractions.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch2\u003eDosage \u0026amp; Administration\u003c\/h2\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eRoute:\u003c\/strong\u003e Papaverine comes as a ready-to-inject solution. It is administered by a doctor or trained nurse via \u003cstrong\u003eintramuscular (IM)\u003c\/strong\u003e or \u003cstrong\u003eslow intravenous (IV)\u003c\/strong\u003e injection. For erectile dysfunction, it is injected \u003cstrong\u003eintracavernosally\u003c\/strong\u003e into the penis (often with local anesthesia).\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eTypical Dose:\u003c\/strong\u003e A single 2 mL vial (60 mg) is a common dose. The exact regimen (frequency and duration) is determined by the prescribing physician based on the indication. For ED therapy, injections are often given 1–3 times per week as needed. For vascular or spasm uses, a single injection or infusion may be done daily or every few days as prescribed.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eInjection Technique:\u003c\/strong\u003e Always inject \u003cstrong\u003eslowly\u003c\/strong\u003e over 1–2 minutes to avoid cardiovascular side effects. Rapid IV injection can cause serious arrhythmias or respiratory arrest, so careful administration is critical. After injection, the patient should be monitored briefly for any immediate reactions.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eAdministration Setting:\u003c\/strong\u003e Because of the risk of cardiovascular effects and the need for sterility, Papaverine injection \u003cstrong\u003emust only be used under medical supervision\u003c\/strong\u003e. It is not a self-injectable medication. Patients should lie down or sit during injection to reduce risk of fainting from hypotension.\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003ePrecautions:\u003c\/strong\u003e Prior to administration, the doctor will review the patient’s health history. Inform your healthcare provider about any heart conditions (arrhythmias, heart block), blood pressure issues, liver problems, or other medications. Those conditions may require dose adjustments or extra monitoring.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch2\u003eStorage \u0026amp; Handling\u003c\/h2\u003e\n\u003cp\u003eEach ampoule is single-use. Store Papaverine Injection vials at room temperature \u003cstrong\u003ebelow 30 °C\u003c\/strong\u003e, away from direct sunlight. Do not freeze. Keep the ampoules in the original box until use to protect from light. After opening, do not save any leftover; dispose of used vials properly. Always check the solution before use – it should be clear and free of particles. If the ampoule is damaged or the solution is discolored, do not use it.\u003c\/p\u003e\n\u003ch2\u003eSide Effects \u0026amp; Precautions\u003c\/h2\u003e\n\u003cp\u003e\u003cstrong\u003eCommon Side Effects (IV\/IM use)\u003c\/strong\u003e – Patients may experience mild to moderate side effects due to vasodilation or muscle relaxation. These include: nausea, headache, flushing of the face, sweating, abdominal discomfort, mild hypotension (low blood pressure), dizziness, and local injection site irritation. Usually these symptoms are transient.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eCardiovascular Risks\u003c\/strong\u003e – Because Papaverine lowers vascular resistance, it can \u003cstrong\u003edrop blood pressure\u003c\/strong\u003e. Rapid IV injection especially risks serious arrhythmias or cardiac events. For safety, infusion should be very slow and the patient monitored. In rare cases, IV use has caused arrhythmias, apnea, or thrombophlebitis at the injection site.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003eED Therapy Risks\u003c\/strong\u003e – With penile injection, the most concerning risk is \u003cstrong\u003epriapism\u003c\/strong\u003e: a prolonged, painful erection lasting \u0026gt;4 hours. Patients must be counseled to seek immediate medical help if an erection persists, as this is an emergency. Long-term intracavernosal use can also rarely lead to fibrosis (scar tissue) in the penis.\u003c\/p\u003e\n\u003cp\u003e\u003cstrong\u003ePrecautions:\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cem\u003eHeart Conditions:\u003c\/em\u003e Contraindicated in complete heart block or severe bradycardia. Use with caution in any patient with conduction disorders or on antiarrhythmic drugs.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003eBlood Pressure:\u003c\/em\u003e Patients on antihypertensives or those prone to hypotension should be monitored closely, as Papaverine can amplify blood pressure-lowering effects.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003eOther Medications:\u003c\/em\u003e Inform your doctor of all drugs you take; interactions are possible. For example, combining with other vasodilators or nitrates could cause excessive hypotension.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003eAllergy:\u003c\/em\u003e Do not use if allergic to papaverine or opium derivatives.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003ePregnancy \u0026amp; Breastfeeding:\u003c\/em\u003e Classified \u003cstrong\u003ePregnancy Category C\u003c\/strong\u003e. Use only if clearly needed and if benefits outweigh risks. It is excreted in breast milk, so nursing mothers should exercise caution.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003eDependence:\u003c\/em\u003e Long-term use can cause drug dependence. Use only for the prescribed duration.\u003c\/li\u003e\n\u003cli\u003e\n\u003cem\u003eSide Effects Management:\u003c\/em\u003e Dizziness or drowsiness may occur; avoid driving or operating machinery until you know how Papaverine affects you. Drink water if feeling faint. Report severe symptoms (chest pain, irregular heartbeat, severe nausea) to a doctor immediately.\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cspan class=\"VODHU pdMy8\"\u003eIn summary, Papaverine 60mg\/2mL single-dose injection is a \u003cstrong\u003epharmacy-grade medication\u003c\/strong\u003e with strong vasodilatory and antispasmodic action. Under medical supervision, it provides targeted relief for circulation and muscle spasm disorders. Always use it exactly as directed by your healthcare provider to maximize benefits and minimize risks.\u003c\/span\u003e\u003c\/p\u003e","brand":"Oryza Pharmaceuticals","offers":[{"title":"Default Title","offer_id":53871120023920,"sku":"72516-0024-10","price":465.0,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/files\/Papaverine-Hydrochloride-Injection-60-mg-Muscle-Relaxant.jpg?v=1780665007"}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0996\/0350\/collections\/Muscle_Relaxants.jpg?v=1733412985","url":"https:\/\/www.mountainside-medical.com\/collections\/muscle-relaxants.oembed?constraint=smooth-muscles","provider":"Mountainside Medical","version":"1.0","type":"link"}